X-Message-Number: 30106 Date: Thu, 6 Dec 2007 09:44:47 -0800 (PST) From: Subject: types of cryoprotectant toxicity Part 1 [Cryoprotectant dependant toxicity can be divided in three types of damage: osmotic, intrinsic, and extrinsic. Osmotic damage occurs when cells shrink too much, after being exposed to too high a concentration of permeating cryoprotectants too quickly. An effective means for completely eliminating this type of damage, is to reduce the rate of increase in the molarity of cryoprotectants, so cells never shrink beyond a certain threshold, which will vary by cell type. In the addition to direct cellular shrinkage, indirect shrinkage can be triggered by an intact blood/brain barrier, which can allow water to pass out of the brain too quickly, while cryoprotectants only slowly enter the brain to replace the lost fluid. Unfortunately the price paid for gradually ramping up molarity, is increased length of time of exposure to cryoprotectants, which can in turn increase both intrinsic as well as extrinsic toxicity. The addition of small amounts of rapidly permeating methanol has been used to limit osmotic damage. Intrinsic damage is time dependant direct damage to cellular constituents by concentrations of cryprotectants beyond a certain threshold. Examples of intrinsic damage include high molar propylene glycol destabilizing cell membranes, while DMSO, and formamide directly denature DNA. Intrinsic damage can be effectively eliminated by reducing the period of exposure. Such rapid freezing techniques can work for individual cells, but are impossible to impliment for organ systems, due to the prolonged period of time required for cryoprotectant equilibration, as well as high thermal inertia. However not all cryoprotectants show significant intrinsic toxicity. Glycerol appears to be virtually free of this type of toxicity, with ethylene glycol in second place. However glycerol only slowly diffuses across cell membranes, and so greatly increases the risk of osmotic damage. Ethylene glycol's major limitation is in the area of extrinsic toxicity. Extrinsic toxicity is time dependant damage to cellular constituents by either metabolites of cryoprotectants, or to free radicals generated during the process of their metabolism. Extrinsic damage can be eliminated by blocking metabolism of cryoprotectants. For example cooling from room temperature tends to reduce metabolism, and thereby helps to limit this type of damage. There are other options to reduce metabolism of cryoprotectants such as inhibiting an enzyme called alcohol dehydrogenase. The main destructive metabolite of ethylene glycol is known to be calcium oxalate. Ethanol has been used to reduce the metabolism of ethylene glycol. IMHO, the reason ethylene glycol has seen use in vitrification solutions despite a high extrinsic toxicity may be due to a similar reduction of ethylene glycol metabolism by the other cryoprotectants.] Rate This Message: http://www.cryonet.org/cgi-bin/rate.cgi?msg=30106