X-Message-Number: 4805 Date: Tue, 22 Aug 1995 19:48:43 +0200 (MET DST) From: Eugene Leitl <> Subject: fixation =-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-= Also in context of concurrent aldehyde/polyol perfusion: "Avanced Organic Chemistry - Reactions, Mechanisms and Structure", Jerry March, 3rd ed., John Wiley & Sons (1985), pp 789-791. 6-6 The Addition of Alcohols to Aldehyds and Ketones (Dialkoxy-de-oxo-bisubstitution) [picture] Acetals and ketals are formed by treatment of aldehydes and ketones, respectively, with alcohols in the presence of acid catalysts. This is a reversible reaction, and acetal and ketals can be hydrolyzed by treatment with acid (0-7). With small ^^^^^^^^^^ unbranched aldehydes the equilibrium lies to the right. If it ^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^ [my emphasis] is desired to prepare ketals, or acetals of larger molecules, the equilibrium must be shifted, usually by removal of water. This can be done by azeotropic destillation, ordinary destillation, or the uses of a drying agent such as Al_2O_3 or a molecular sieve. The reaction in neither direction is catalyzed by bases, so most acetals and ketals are quite stable to bases, though they are easily hydrolyzed by acids. This makes this reaction a useful method of protection of aldehyde or ketone functions from attack by bases. The reaction is of wide scope. Most aldehydes are easily converted to acetals. With ketones the process is more difficult, presumably by steric reasons, and the reaction often fails, though many ketals, especially from cyclic ketones, have been made in this manner. Many functional groups can be presented without being affected. 1,2-Glycols and 1,3-glycols form cyclic acetals and ketals, e.g. [picture] and these are often used to protect aldehydes and ketones. [ Especially crosslinking agents' (as methanal) reactivity is vastly enhanced due to occurence intermolecular reactions (entropy favoured) with the polyol :( -- Eugene ] =-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-= "Techniques in Immunocytochemistry", Vol 1., Gillian R. Bullock, Peter Petrusz, Edit., Academic Press, Inc. (London) Ltd. (1982). "Tissue Preparation Methods for Immunochemistry", Per Brantzaeg, pp. 2-75. "The Protein A-Gold (pAg) Technique - A Qualitative and Quantitative Approach for Antigen Localization on Thin Sections", J"urgen Roth, pp. 108-133. "Light Microscopic Immunocytochemistry with Fixed, Unembedded Tissues", Reinhard Grzanna, pp. 183-204. =-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-= Tissue Preparation Methods for Immunochemistry. I. Introduction [...] The purpose of fixation is, in immunochemical terms, to arrest enzymatic activity sufficiently rapidly to avoid structural decomposition, to hinder diffusion of peptides and proteins into and out of cells, and to fortify the tissue against deletorious effects during the various stages in the preparation of sections. Artifacts may develop when the tissue specimens are subjected to dehydration, clearing and embedding, and when the sections are being cut, floated, stretched, dried, dewaxed, rinsed, incubated, and washed. In addition, structural decomposition and diffusion artefacts my develop before the fixation process takes place - either in vivo because of denaturation or necrosis of cells, or in vitro because of autolysis, osmotic damage, drying, or rough mechanical treatment. [...] II. Principles of Tissue Preparation A. Fixation Methods Although fixation is necessary to avoid artefactual difussion of soluble tissue components and decomposition of structures, it constitutes in itself a major artefact since the living cell and surroundings are fluid or semi-fluid in nature. A detailed description of different fixatives and their action on various tissue components can be found in several major texts on histochemistry and hisopathology (Culling, 1974; Lillie and Fullmer, 1976; Nairn, 1976; Pearse 1980). Fixatives such as ethanol and methanol immobilize proteins and carbohydrates by precipitation. The denaturing effect of these fixatives is relatively mild and to large extent reversible. Thus, proteins may be redissolved in a fairly native state after ethanol fixation. It follows that adequate immobilization of antigens in tissue sections is far from guaranteed. Moreover, dehydration takes place simultaneously with the fixation process so that morphological preservation may be unsatisfactory due to shrinkage. Immobilization of peptides and proteins is best afforded by bifunctional cross-linking fixatives such as formaldehyded and glutaraldehyde, which also preserve more adequately the structures of cells and tissue. However, cross-linking necessarily leads to more severe antigen denaturation than precipitation; this particularly so for large protein antigenes whose reactivity does not depend on primary structure alone but also on conformational features (Kauzmann, 1959). Even the antigenicity of peptides is adversely affected by the aldehyde-based fixatives which react with primary amino groups, and several alternative cross-linking agents have been suggested for the localization of peptide hormones. These fixatives include water-soluble carbodiimide (Kendall et al., 1971) and the bifunctional reagent parabenzoquinone (Pearse and Polak, 1975). Several variables will influence the effect of cross-linking fixatives on antigenicity. Thus, when formaldehyde is used the number of methylene bridges formed depends not only on the concentrations of the fixative, but also on the temperature, pH and time of exposure. The deletorious effect on antigen reactivity may be partially reversed before tissue eembedding by extensive washing in water or treeatment with sucrose (Eidelman and Berschauer, 1969; Deng and Beutner, 1974). The aldehyde-based fixatives induce both intermolecular and intramolecular bridges. Due to such extensive formation of cross-linkage formaldehyde, and even more so glutaraldehyde, may in addition to denaturation may cause masking of antigens by steric hindrance. This phenomenon is pronounced when the actual antigen is mixed with high concentrations of other proteins (Rognum et al., 1980; Hed and Enestrom, 1981). The suggestions made by some authors (Sternberger, 1979) that the deletorious effects of aldehyde-based fixatives can be compensated for by use of a highly sensitive immunohistochemical method is thus only partially true. It is necessary to take into account that an uneven antigen masking takes place according to location; interpretation of any observed antigen distribution can only be meaningful if this fact is kept in mind, regardless of whether immunofluorescence or immunoenzyme methods are used for detection. B. Exposure of Hidden Antigens [ various immunostain enhancement procedures ] C. Unmasking of Antigens Concealed During Fixation [ using proteolytic digestion ] D. Removal of Diffusible Proteins Before Fixation [ discerning diffusible from membrane-bound/aggregated antigens ] E. Pre-fixation Diffusion Artefacts A problem that has received little attention, both in immunobiological and immunopathological studies, is the fact that immunoglobulins and complement factor C3 are present in interstital fluid in relatively high concentrations and may, therefore, enter cells by passive diffusion (Mason and Biberfeld, 1980; Mason et al., 1980; Brandtzaeg, 1981b). Cells subjected to such uptake often appear morphologically intact; only slight plasma membrane damage may thus have been induced prior to fixation, either in vivo or in vitro. Rough treatment of the tissue specimen and retarded fixation contribute to this aftefact. Kent (1966, 1967) showed that uptake of plasma proteins in ischaemic myocardium occured according to the size of the molecules and the degree of injury. In squamous epithelia superficial degenerating cells commonly contain plasma proteins in quantitaive proportions corresponding to the content found in the underlying connective tissue (Brandtzaeg and Kraus, 1965; Brandtzaeeg, 1975; Brandtzaeg et al. 1978). Leakage of plasma proteins into columnar epithelium has likewise been described (Mason and Piris, 1980). [...] F. Post-fixation Diffusion Artefacts It was pointed out above (Section II.A) that even large protein anntigens may not always be sufficiently immobilized by ethanol fixation to avoid their dissolution during incubation and washing of the tissue section. We encountered this artifact in immunofluorscence staining experiments when we prolonged the incubation with fluorochrome conjugates from 30 min 20 h (Brandtzaeg, 1981b). A decreased staining intensity could bee ascribed both to loss of antigen and to partial neutralization of the conjugate during the prolonged incubation time, especially in the central areas of the section. This problem may be even greater when working with unfixed or lighly fixed cryostat sections. [...] G. Conclusion Ethanol acts as a fixative by protein precipitation whereas formaldehyde immobilizes the proteins by the formation of cross-linkages (Fig. 19). Immobilization of small antigens, such as peptide hormones, can only be obtained safely with some kind of cross-bridging fixative, and their antigenicity is relatively well preserved by this procedure. The antigenicity of protein antigens, an the other hand, does not depend on the primary structure alone but also on conformational features, which may be severely altered by the fixation process. Due to extensive formation of cross-linkages, aldehyde-based fixatives produce and additional artifact, namely masking of antigens - particularly those mixed with high concentrations of other proteins. [...] III. Immunochemical Testing of Fixatives A. Artificial Test Substrates [...] B. Performance Testing on Biological Substrates [...] 1. Routine Formalin Fixation [...] 2. Glutaraldehyde-Formaldehyde Glutaraldehyde is a dialdehyde and has a much greater cross-linking potential than formaldehyde. Our tests with artificial substrates showed that fixation with a combination of 1 percent glutaraldehyde and 3.5 percent formaldehyde yielded somewhat reduced detection sensivity for IgG comparted with routine formalin fixation, and the masking was even more pronounced at high antigen concentraions (Fig. 23). Despite this properties, glutaraldehyde-containing fixatives have been preferred in several studies based on PAP staining (Sternberger, 1979). A significant advantage of the glutaraldehyde-formaldehyde combination is that it gives satisfactory preservation of tissue both for routine histological staining methods and for electron microscopical studies (McDowell and Trump, 1976). [...] 3. Baker's Formol Calcium This fixative has been recommended for the preservation of phospholipids in tissues. Our results with fixation of IgG and IgA in artificial substrates indicated that Baker's formol calcium yielded somewhat better detection sensitivity and much less cross-bridging of protein than the other aldehyde-based fixatives (Fig. 23). [...] 4. Formol Sublimate [ several ugly mercuric chloride + additives preparations ] 5. Acetic Acid-Formol Saline [...] Acetic acid-formol saline thus seems to be the aldehyde-based fixative of choice for intracellular protein antigens when proteolytic digestion of tissue section is undesirable. However, this fixative does not permit the study of extracellular or membrane-associated antigens. The results of Curran and Gregory (1980) indicated that it is the low pH of the formaldehyde solution rather than the acetic acid per se that explains the favourable results. 6. Bouin's Fluid This fixative is known to penetrate rapidly and to cause little shrinkage. In addition to formaldehyde and acetic acid, it contains picric acid, which precipitates proteins and combines with them to form picrates and also produces intermolecular salt links (Pearse, 1980). [...] 7. Susa Fixative This fixative has properties similiar tot Bouin's fluid, but contains trichloroacetic acid and mercuric chloride instead of picric acid. [...] Alltogether, there were no apparent advantages in using Susa fixative for immunochemistry of immunoglobulins. 8. Carbodiimide Water-soluble carbodiimides have been widely used to prepare immunogenic conjugates by coupling small peptides to carrier proteins. They effect polymerization by initial attack of carboxyl groups to give an acylisourea, which next may react with an adjacent amino group to crosslink through an amide bond (Stark, 1970). A requirement for cross-linking, therefore, is probably close proximity between carboxyl and amino groups; this may explain that although carbodiimides are as efficient as aldehydes for insolubilization of proteins (Yamamoto and Yasuda, 1977), we found substantially less masking of antigenicity after tissue fixation with the former (Brandtzaeg and Rognum, 1982a,b). [...] Carbodiimide is thus a cross-linking fixative that for protein antigens gives a result similiar to that obtained after ethanol fixation (Fig. 23). It has recently been shown that the cytosol matrix remains permeable after fixation with carbodiimide even when 0.3 percent glutaraldehyde is addd to it (Willingham and Yamada, 1979). This combination enhances morphological preservation and offers promises for application in immunoelectron microscopical localization studies. [ On the whole carbodiimides might be promising auxiliary perfusion agents, particularly since they do not react with polyols but require carboxyl/amine group for a crosslink. Of course, their influence on perfusion (blood-brain barrier) has to be checked first. Membrane-shuttle agents might be instrumental here, albeit artefacting on their own rights -- Eugene ] 9. Ethanol The Sainte-Marie (1962) cold ethanol-fixation procedure afforded superior detection sensitivity for IgG and IgA in artificial substrates, and superior immunofluorescence staining intensity for epithelial SC and IgA (Fig. 23). The same held true for immunoglobulin-producing cells of all isotypes when the prefixation washing step was included (Section II. D), and for intracellular J chain when the sections were treated with acid urea (Section II. B). The advantages and drawbacks of tissue preparation methods based on ethanol fixation have been further discussed in Sections II. C, II. E, II.F and II.G and in previous publications (Brandtzaeg, 1974, 1981b). 10. Conclusion [ not much new, here ] IV. Choice of Tissue Preparation Method A. Extracellular and Basement Membrane-Assotiated Protein Antigens [...] B. Cell-Surface and Cytoplasmic Immunoglobulin Components Including J Chain and SC [...] C. Cytoplasmic Enzymes [...] D. Cytoplasmic Hormones [...] E. Miscellaneous Cellular and Tissue Antigens [...] F. Conclusion Tissue preparation is the cornerstone of immunohistochemistry, but is still a subject of much antiquity and ambiguity. There is a need to clarify basic mechanisms rather than to introduce unjustified modifications of existing methods. Furthere progress can only be made when knowledge of the various antigens and their microenvironment is considered together with knowledge of the chemistry of fixation. Statements made in the literature about a general applicability of certain fixatives are likely to be false. It seems that many antigens require a tailor-made tisue preparation technique for optimal preservation and precise localization. From a morphological point of view cross-linking fixatives are generally preferable, but the antigenic masking caused by them is, apparently, a more universal problem in immunohistochemistry than earlier believed. Although proteolytic unmasking to some extent is possible, optimal preservation of antigenicity and morphology is not always compatible with such tretment. It is important that those entering the field of immunohistochemistry be aware of the fact that success is not a matter of mere stain technology in terms of antigen labeling by immunological reactions. The primary and crucial substrate for this reactions is the antigenicity that has been preserved and rendered accessible in the tissue section. In addition comes the goal of adequate morphology. V. Acknowledgements [...] VI. References [...] =-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-= "The Protein A-Gold (pAg) Technique - A Qualitative and Quantitative Approach for Antigen Localization on Thin Sections", J"urgen Roth, pp. 108-133. [...] A. Tissue Fixation In order to obtain adequate immunocytochemical localization of antigens, the fixatives used should stabilize cellular structures to such an extent that artefactual diffusion and replacement of antigenic material or its extraction is prevented and good preservation of cellular fine structure is achieved. On the other hand, the fixative should preserve as much as possible the tertiary structure of antigens to retain a good reactivity with the antibodies. A common phenomenon in post-embedding staining procedures is that excellent structural preservation often results in drastic diminution of antigenicity since fixatives affect fine structure and antigenicity inversely. Therefore, conditions of fixation have to be devised which preserve adequately both cellular fine structure and antigenicity. Among the fixatives used in electron microscopy, aldehydes fulfil these requirements most closely. Other fixatives, such as carboddimide (Polak et al., 1972; Hassel and Hand, 1974; Yamamoto and Yasuda, 1977) and diimidoesters (McLean and Singer, 1970; Ono et al., 1976) have been proposed, but have not been widely tested as yet. Kraehenbuhl et al. (1977) have shown that individual enzymes are affected differently by glutaraldehyde but that low concentrations of glutaraldehyde (0.5 percent) are commensurate with good preservation of both the antigenic properties of pancreatic enzymes and the fine structure of pancreatic tissue. For this reason, we routinely use a 2 h fixation with 0.5 percent glutaraldehyde solution in PBS at room temperature for pancreatic tissue (Bendayan et al., 1980). We also tested fixation with picric acid-formaldehyde solution (Stefanini et al., 1967) which gave a more intense labelling compared to glutaraldehyde fixation but at the expense of fine structural preservation. In our studies on localization of polypeptide hormones we found good preservation of antigenicity after fixation with relatively high concentration of aldehyde (up to 4 percent glutaraldehyde concentration or mixtures of 3 percent glutaraldehyde with 2 percent formaldehyde). Osmium fixation severely influences the antigenicity of many proteins. Only a few antigens have been shown to resist such a fixation protocol (Nakane, 1971; Erlandsen et al., 1979). We observed that aldehyde fixation followed by 1 percent osmium tetroxide fixation for 1 h allowed localization of insulin in pancreatic B cells as in the only aldehyde fixed tissue. On the contrary, we found that aldehyde fixation followed by 1 percent osmium tetroxide for 15 min reduced the labelling intensity for amylase in rat pancreatic tissue by 70 percent. In general, localization of an antigen should be tried first on tissue fixed with 0.5 to 1 percent buffered glutaraldehyde solution since this fixative sufficiently preserves many antigens for subsequent demonstration with the pAg technique. However, for each particular cell type or tissue one has to determine the fixation conditions which are subject: fixation =-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-= Also in context of concurrent aldehyde/polyol perfusion: "Avanced Organic Chemistry - Reactions, Mechanisms and Structure", Jerry March, 3rd ed., John Wiley & Sons (1985), pp 789-791. 6-6 The Addition of Alcohols to Aldehyds and Ketones (Dialkoxy-de-oxo-bisubstitution) [picture] Acetals and ketals are formed by treatment of aldehydes and ketones, respectively, with alcohols in the presence of acid catalysts. This is a reversible reaction, and acetal and ketals can be hydrolyzed by treatment with acid (0-7). With small ^^^^^^^^^^ unbranched aldehydes the equilibrium lies to the right. If it ^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^^ [my emphasis] is desired to prepare ketals, or acetals of larger molecules, the equilibrium must be shifted, usually by removal of water. This can be done by azeotropic destillation, ordinary destillation, or the uses of a drying agent such as Al_2O_3 or a molecular sieve. The reaction in neither direction is catalyzed by bases, so most acetals and ketals are quite stable to bases, though they are easily hydrolyzed by acids. This makes this reaction a useful method of protection of aldehyde or ketone functions from attack by bases. The reaction is of wide scope. Most aldehydes are easily converted to acetals. With ketones the process is more difficult, presumably by steric reasons, and the reaction often fails, though many ketals, especially from cyclic ketones, have been made in this manner. Many functional groups can be presented without being affected. 1,2-Glycols and 1,3-glycols form cyclic acetals and ketals, e.g. [picture] and these are often used to protect aldehydes and ketones. [ Especially crosslinking agents' (as methanal) reactivity is vastly enhanced due to occurence intermolecular reactions (entropy favoured) with the polyol :( -- Eugene ] =-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-= "Techniques in Immunocytochemistry", Vol 1., Gillian R. Bullock, Peter Petrusz, Edit., Academic Press, Inc. (London) Ltd. (1982). "Tissue Preparation Methods for Immunochemistry", Per Brantzaeg, pp. 2-75. "The Protein A-Gold (pAg) Technique - A Qualitative and Quantitative Approach for Antigen Localization on Thin Sections", J"urgen Roth, pp. 108-133. "Light Microscopic Immunocytochemistry with Fixed, Unembedded Tissues", Reinhard Grzanna, pp. 183-204. =-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-= Tissue Preparation Methods for Immunochemistry. I. Introduction [...] The purpose of fixation is, in immunochemical terms, to arrest enzymatic activity sufficiently rapidly to avoid structural decomposition, to hinder diffusion of peptides and proteins into and out of cells, and to fortify the tissue against deletorious effects during the various stages in the preparation of sections. Artifacts may develop when the tissue specimens are subjected to dehydration, clearing and embedding, and when the sections are being cut, floated, stretched, dried, dewaxed, rinsed, incubated, and washed. In addition, structural decomposition and diffusion artefacts my develop before the fixation process takes place - either in vivo because of denaturation or necrosis of cells, or in vitro because of autolysis, osmotic damage, drying, or rough mechanical treatment. [...] II. Principles of Tissue Preparation A. Fixation Methods Although fixation is necessary to avoid artefactual difussion of soluble tissue components and decomposition of structures, it constitutes in itself a major artefact since the living cell and surroundings are fluid or semi-fluid in nature. A detailed description of different fixatives and their action on various tissue components can be found in several major texts on histochemistry and hisopathology (Culling, 1974; Lillie and Fullmer, 1976; Nairn, 1976; Pearse 1980). Fixatives such as ethanol and methanol immobilize proteins and carbohydrates by precipitation. The denaturing effect of these fixatives is relatively mild and to large extent reversible. Thus, proteins may be redissolved in a fairly native state after ethanol fixation. It follows that adequate immobilization of antigens in tissue sections is far from guaranteed. Moreover, dehydration takes place simultaneously with the fixation process so that morphological preservation may be unsatisfactory due to shrinkage. Immobilization of peptides and proteins is best afforded by bifunctional cross-linking fixatives such as formaldehyded and glutaraldehyde, which also preserve more adequately the structures of cells and tissue. However, cross-linking necessarily leads to more severe antigen denaturation than precipitation; this particularly so for large protein antigenes whose reactivity does not depend on primary structure alone but also on conformational features (Kauzmann, 1959). Even the antigenicity of peptides is adversely affected by the aldehyde-based fixatives which react with primary amino groups, and several alternative cross-linking agents have been suggested for the localization of peptide hormones. These fixatives include water-soluble carbodiimide (Kendall et al., 1971) and the bifunctional reagent parabenzoquinone (Pearse and Polak, 1975). Several variables will influence the effect of cross-linking fixatives on antigenicity. Thus, when formaldehyde is used the number of methylene bridges formed depends not only on the concentrations of the fixative, but also on the temperature, pH and time of exposure. The deletorious effect on antigen reactivity may be partially reversed before tissue eembedding by extensive washing in water or treeatment with sucrose (Eidelman and Berschauer, 1969; Deng and Beutner, 1974). The aldehyde-based fixatives induce both intermolecular and intramolecular bridges. Due to such extensive formation of cross-linkage formaldehyde, and even more so glutaraldehyde, may in addition to denaturation may cause masking of antigens by steric hindrance. This phenomenon is pronounced when the actual antigen is mixed with high concentrations of other proteins (Rognum et al., 1980; Hed and Enestrom, 1981). The suggestions made by some authors (Sternberger, 1979) that the deletorious effects of aldehyde-based fixatives can be compensated for by use of a highly sensitive immunohistochemical method is thus only partially true. It is necessary to take into account that an uneven antigen masking takes place according to location; interpretation of any observed antigen distribution can only be meaningful if this fact is kept in mind, regardless of whether immunofluorescence or immunoenzyme methods are used for detection. B. Exposure of Hidden Antigens [ various immunostain enhancement procedures ] C. Unmasking of Antigens Concealed During Fixation [ using proteolytic digestion ] D. Removal of Diffusible Proteins Before Fixation [ discerning diffusible from membrane-bound/aggregated antigens ] E. Pre-fixation Diffusion Artefacts A problem that has received little attention, both in immunobiological and immunopathological studies, is the fact that immunoglobulins and complement factor C3 are present in interstital fluid in relatively high concentrations and may, therefore, enter cells by passive diffusion (Mason and Biberfeld, 1980; Mason et al., 1980; Brandtzaeg, 1981b). Cells subjected to such uptake often appear morphologically intact; only slight plasma membrane damage may thus have been induced prior to fixation, either in vivo or in vitro. Rough treatment of the tissue specimen and retarded fixation contribute to this aftefact. Kent (1966, 1967) showed that uptake of plasma proteins in ischaemic myocardium occured according to the size of the molecules and the degree of injury. In squamous epithelia superficial degenerating cells commonly contain plasma proteins in quantitaive proportions corresponding to the content found in the underlying connective tissue (Brandtzaeg and Kraus, 1965; Brandtzaeeg, 1975; Brandtzaeg et al. 1978). Leakage of plasma proteins into columnar epithelium has likewise been described (Mason and Piris, 1980). [...] F. Post-fixation Diffusion Artefacts It was pointed out above (Section II.A) that even large protein anntigens may not always be sufficiently immobilized by ethanol fixation to avoid their dissolution during incubation and washing of the tissue section. We encountered this artifact in immunofluorscence staining experiments when we prolonged the incubation with fluorochrome conjugates from 30 min 20 h (Brandtzaeg, 1981b). A decreased staining intensity could bee ascribed both to loss of antigen and to partial neutralization of the conjugate during the prolonged incubation time, especially in the central areas of the section. This problem may be even greater when working with unfixed or lighly fixed cryostat sections. [...] G. Conclusion Ethanol acts as a fixative by protein precipitation whereas formaldehyde immobilizes the proteins by the formation of cross-linkages (Fig. 19). Immobilization of small antigens, such as peptide hormones, can only be obtained safely with some kind of cross-bridging fixative, and their antigenicity is relatively well preserved by this procedure. The antigenicity of protein antigens, an the other hand, does not depend on the primary structure alone but also on conformational features, which may be severely altered by the fixation process. Due to extensive formation of cross-linkages, aldehyde-based fixatives produce and additional artifact, namely masking of antigens - particularly those mixed with high concentrations of other proteins. [...] III. Immunochemical Testing of Fixatives A. Artificial Test Substrates [...] B. Performance Testing on Biological Substrates [...] 1. Routine Formalin Fixation [...] 2. Glutaraldehyde-Formaldehyde Glutaraldehyde is a dialdehyde and has a much greater cross-linking potential than formaldehyde. Our tests with artificial substrates showed that fixation with a combination of 1 percent glutaraldehyde and 3.5 percent formaldehyde yielded somewhat reduced detection sensivity for IgG comparted with routine formalin fixation, and the masking was even more pronounced at high antigen concentraions (Fig. 23). Despite this properties, glutaraldehyde-containing fixatives have been preferred in several studies based on PAP staining (Sternberger, 1979). A significant advantage of the glutaraldehyde-formaldehyde combination is that it gives satisfactory preservation of tissue both for routine histological staining methods and for electron microscopical studies (McDowell and Trump, 1976). [...] 3. Baker's Formol Calcium This fixative has been recommended for the preservation of phospholipids in tissues. Our results with fixation of IgG and IgA in artificial substrates indicated that Baker's formol calcium yielded somewhat better detection sensitivity and much less cross-bridging of protein than the other aldehyde-based fixatives (Fig. 23). [...] 4. Formol Sublimate [ several ugly mercuric chloride + additives preparations ] 5. Acetic Acid-Formol Saline [...] Acetic acid-formol saline thus seems to be the aldehyde-based fixative of choice for intracellular protein antigens when proteolytic digestion of tissue section is undesirable. However, this fixative does not permit the study of extracellular or membrane-associated antigens. The results of Curran and Gregory (1980) indicated that it is the low pH of the formaldehyde solution rather than the acetic acid per se that explains the favourable results. 6. Bouin's Fluid This fixative is known to penetrate rapidly and to cause little shrinkage. In addition to formaldehyde and acetic acid, it contains picric acid, which precipitates proteins and combines with them to form picrates and also produces intermolecular salt links (Pearse, 1980). [...] 7. Susa Fixative This fixative has properties similiar tot Bouin's fluid, but contains trichloroacetic acid and mercuric chloride instead of picric acid. [...] Alltogether, there were no apparent advantages in using Susa fixative for immunochemistry of immunoglobulins. 8. Carbodiimide Water-soluble carbodiimides have been widely used to prepare immunogenic conjugates by coupling small peptides to carrier proteins. They effect polymerization by initial attack of carboxyl groups to give an acylisourea, which next may react with an adjacent amino group to crosslink through an amide bond (Stark, 1970). A requirement for cross-linking, therefore, is probably close proximity between carboxyl and amino groups; this may explain that although carbodiimides are as efficient as aldehydes for insolubilization of proteins (Yamamoto and Yasuda, 1977), we found substantially less masking of antigenicity after tissue fixation with the former (Brandtzaeg and Rognum, 1982a,b). [...] Carbodiimide is thus a cross-linking fixative that for protein antigens gives a result similiar to that obtained after ethanol fixation (Fig. 23). It has recently been shown that the cytosol matrix remains permeable after fixation with carbodiimide even when 0.3 percent glutaraldehyde is addd to it (Willingham and Yamada, 1979). This combination enhances morphological preservation and offers promises for application in immunoelectron microscopical localization studies. [ On the whole carbodiimides might be promising auxiliary perfusion agents, particularly since they do not react with polyols but require carboxyl/amine group for a crosslink. Of course, their influence on perfusion (blood-brain barrier) has to be checked first. Membrane-shuttle agents might be instrumental here, albeit artefacting on their own rights -- Eugene ] 9. Ethanol The Sainte-Marie (1962) cold ethanol-fixation procedure afforded superior detection sensitivity for IgG and IgA in artificial substrates, and superior immunofluorescence staining intensity for epithelial SC and IgA (Fig. 23). The same held true for immunoglobulin-producing cells of all isotypes when the prefixation washing step was included (Section II. D), and for intracellular J chain when the sections were treated with acid urea (Section II. B). The advantages and drawbacks of tissue preparation methods based on ethanol fixation have been further discussed in Sections II. C, II. E, II.F and II.G and in previous publications (Brandtzaeg, 1974, 1981b). 10. Conclusion [ not much new, here ] IV. Choice of Tissue Preparation Method A. Extracellular and Basement Membrane-Assotiated Protein Antigens [...] B. Cell-Surface and Cytoplasmic Immunoglobulin Components Including J Chain and SC [...] C. Cytoplasmic Enzymes [...] D. Cytoplasmic Hormones [...] E. Miscellaneous Cellular and Tissue Antigens [...] F. Conclusion Tissue preparation is the cornerstone of immunohistochemistry, but is still a subject of much antiquity and ambiguity. There is a need to clarify basic mechanisms rather than to introduce unjustified modifications of existing methods. Furthere progress can only be made when knowledge of the various antigens and their microenvironment is considered together with knowledge of the chemistry of fixation. Statements made in the literature about a general applicability of certain fixatives are likely to be false. It seems that many antigens require a tailor-made tisue preparation technique for optimal preservation and precise localization. From a morphological point of view cross-linking fixatives are generally preferable, but the antigenic masking caused by them is, apparently, a more universal problem in immunohistochemistry than earlier believed. Although proteolytic unmasking to some extent is possible, optimal preservation of antigenicity and morphology is not always compatible with such tretment. It is important that those entering the field of immunohistochemistry be aware of the fact that success is not a matter of mere stain technology in terms of antigen labeling by immunological reactions. The primary and crucial substrate for this reactions is the antigenicity that has been preserved and rendered accessible in the tissue section. In addition comes the goal of adequate morphology. V. Acknowledgements [...] VI. References [...] =-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-= "The Protein A-Gold (pAg) Technique - A Qualitative and Quantitative Approach for Antigen Localization on Thin Sections", J"urgen Roth, pp. 108-133. [...] A. Tissue Fixation In order to obtain adequate immunocytochemical localization of antigens, the fixatives used should stabilize cellular structures to such an extent that artefactual diffusion and replacement of antigenic material or its extraction is prevented and good preservation of cellular fine structure is achieved. On the other hand, the fixative should preserve as much as possible the tertiary structure of antigens to retain a good reactivity with the antibodies. A common phenomenon in post-embedding staining procedures is that excellent structural preservation often results in drastic diminution of antigenicity since fixatives affect fine structure and antigenicity inversely. Therefore, conditions of fixation have to be devised which preserve adequately both cellular fine structure and antigenicity. Among the fixatives used in electron microscopy, aldehydes fulfil these requirements most closely. Other fixatives, such as carboddimide (Polak et al., 1972; Hassel and Hand, 1974; Yamamoto and Yasuda, 1977) and diimidoesters (McLean and Singer, 1970; Ono et al., 1976) have been proposed, but have not been widely tested as yet. Kraehenbuhl et al. (1977) have shown that individual enzymes are affected differently by glutaraldehyde but that low concentrations of glutaraldehyde (0.5 percent) are commensurate with good preservation of both the antigenic properties of pancreatic enzymes and the fine structure of pancreatic tissue. For this reason, we routinely use a 2 h fixation with 0.5 percent glutaraldehyde solution in PBS at room temperature for pancreatic tissue (Bendayan et al., 1980). We also tested fixation with picric acid-formaldehyde solution (Stefanini et al., 1967) which gave a more intense labelling compared to glutaraldehyde fixation but at the expense of fine structural preservation. In our studies on localization of polypeptide hormones we found good preservation of antigenicity after fixation with relatively high concentration of aldehyde (up to 4 percent glutaraldehyde concentration or mixtures of 3 percent glutaraldehyde with 2 percent formaldehyde). Osmium fixation severely influences the antigenicity of many proteins. Only a few antigens have been shown to resist such a fixation protocol (Nakane, 1971; Erlandsen et al., 1979). We observed that aldehyde fixation followed by 1 percent osmium tetroxide fixation for 1 h allowed localization of insulin in pancreatic B cells as in the only aldehyde fixed tissue. On the contrary, we found that aldehyde fixation followed by 1 percent osmium tetroxide for 15 min reduced the labelling intensity for amylase in rat pancreatic tissue by 70 percent. In general, localization of an antigen should be tried first on tissue fixed with 0.5 to 1 percent buffered glutaraldehyde solution since this fixative sufficiently preserves many antigens for subsequent demonstration with the pAg technique. However, for each particular cell type or tissue one has to determine the fixation conditions which are compatible with adequate preservation of fine structure and antigenicity. =-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-=-= Rate This Message: http://www.cryonet.org/cgi-bin/rate.cgi?msg=4805